Contents

Russian Journal of Bioorganic Chemistry


Vol. 48, No. 5, 2022


Pyrazine Derivatives—Versatile Scaffold

N. Tambat, S. K. Mulani, A. Ahmad, S. B. Shaikh and K. Ahmed p. 865  abstract

Hyaluronan Metabolism and Tumor Progression

I. I. Khegai p. 896  abstract

Synthesis, Antiviral, and Antibacterial Activity of the Glycyrrhizic Acid and Glycyrrhetinic Acid Derivatives

E. A. H. Mohammed, Y. Peng, Z. Wang, X. Qiang and Q. Zhao p. 906  abstract

Recent Advances in Protein Kinase CK2, a Potential Therapeutic Target in Cancer

V. B. Nipun and K. A. Amin p. 919  abstract

Influence of the Lipid Moiety Structure on the Insertion/Release of Glycolipids in/from the Cell: A Study with Synthetic Analogs

E. V. Slivka, A. B. Tuzikov, S. V. Khaidukov, V. A. Komarova, S. M. Henry, N. V. Bovin and E. M. Rapoport p. 932  abstract

Synthetic Antimicrobial Peptides: IV. Effect of Cationic Groups of Lysine, Arginine, and Histidine on Antimicrobial Activity of Peptides with a ‘Circular’ Type of Amphipathicity

N. V. Amirkhanov, A. V. Bardasheva, N. V. Tikunova and D. V. Pyshnyi p. 937  abstract

SwissADME Predictions of Drug-Likeness of 5-Nitro Imidazole Derivatives as Potential Antimicrobial and Antifungal Agents

P. Pattanayak p. 949  abstract

Drug Repurposing to Discover Novel Anti-Inflammatory Agents Inhibiting JAK3/STAT Signaling

S. Y. Sheikh, F. Hassan, M. F. Khan, T. Ahamad, W. A. Ansari, Y. Akhter, El-Sayed Khafagy, A. R. Khan and M. Nasibullah p. 958  abstract

Bioinformatics Study of Pioglitazone Analogues as Potential Anti-Diabetic Drugs

Priyaranjini Rao, Ashwini S, Ghazala Masood, Raviraj Kusanur, Vidya Niranjan and Swarna M. Patra p. 976  abstract

Diacylhydrazine Derivatives of 2-(5-(Pyridin-3-yl)-2H-Tetrazol-2-yl)Acetohydrazide and 2-(5-(Pyridin-4-yl)-2H-Tetrazol-2-yl)Acetohydrazide as Potential Inhibitors of Nucleotide Pyrophosphatase

M. Arif, G. Shabir, S. A. Ejaz, A. Saeed, S. U. Khan, J. Lecka, J. Sévigny and J. Iqbal p. 990  abstract

Radioligand Binding Assay for the Simultaneous Determination of β1- and β2-Adrenergic Receptors in Human Blood Cells

A. Y. Shevelev, N. M. Kashirina, L. N. Lipatova, E. V. Yanushevskaya, M. M. Peklo, I. N. Rybalkin, P. N. Rutkevich, O. K. Chusovitina, N. A. Skoblova, Yu. S. Skoblov, T. N. Vlasik and K. A. Zykov p. 1002  abstract

Synthesis and Evaluation of 1,3-Dimethylbarbituric Acid Based Enamine Derivatives as Anti-Alzheimer Agent

S. F. Shaikh, J. J. Uparkar, G. S. Pavale and M. M. V. Ramana p. 1011  abstract

Synthesis of the Antagonist of the GalR2 Galanin Receptor and Studies of Its Biological Activity in Ischemia and Reperfusion of the Rat Heart In Vivo

M. V. Sidorova, M. E. Palkeeva, D. V. Avdeev, I. M. Studneva, L. I. Serebryakova, O. M. Veselova, I. V. Dobrokhotov, A. S. Molokoedov and O. I. Pisarenko p. 1020  abstract

The Synthesis and Anti-inflammatory Studies of New Pyrimidine Derivatives, Inhibitors of Cyclooxygenase Isoforms

Y. Z. Khazimullina, A. R. Gimadieva, V. R. Khairullina, L. F. Zainullina, Y. V. Vakhitova and A. G. Mustafin p. 1027  abstract

Photocaged Small Interfering RNA

E. A. Akhmetova, D. V. Kim, A. S. Dome, M. I. Meschaninova and D. S. Novopashina p. 1036  abstract

Synthesis, Antioxidant, and Antibacterial Activities of Two Novel Series of 3,5-Disubstituted Isoxazole Ether-Linked Isoxazolines and 3,5-Disubstituted Pyrazole Ether-Linked Isoxazolines Mediated by Chloramine-T

E. A. M. Saleh, S. Y. Kotian, A. M. Al Dawsari, I. Hassan, K. Husain, P. C. Abishad, K. Byrappa, R. S. S. AL Sharabi and K. M. L. Rai p. 1043  abstract

Synthesis of Isatin-Based Oxo-Spiro Chromene Schiff’s Bases as Antibacterial and Anticancer Agents

S. N. Dandekar, O. A. Lotlikar, M. M. V. Ramana and S. V. Rathod p. 1053  abstract

Synthesis and β-Lactamase Inhibition Activity of Imidates of Diazabicyclooctane

Lijuan Zhai, Jian Sun, Jingwen Ji, Lili He, Yuanyu Gao, Jinbo Ji, Yuanbai Liu, Yangxiu Mu, Xueqin Ma, Dong Tang, Haikang Yang, Zafar Iqbal and Zhixiang Yang p. 1059  abstract

Synthesis, Characterization, Biological, and Molecular Docking Studies of (Z)-N-Substituted-4-(Pyridin-2-yl)-6-(1H-Pyrrolo[2,3-b]Pyridin-4-yl)Pyrimidin-2-Amine

M. Arshad and M. S. Akhter p. 1068  abstract

Design, Synthesis, Characterization, DFT Calculations, Molecular Docking Study, and Antimicrobial Activity of Hydrazones Bearing Pyrimidine and Sugar Moieties

A. Z. Omar, N. G. A. El-Aleem, S. M. A. Megid and A. A. El-Bardan p. 1076  abstract

Design, Synthesis, and Antitumor Activity Evaluation of 2,4,6-Trisubstituted Quinazoline Derivatives Containing Acrylamide

D. Honglin, G. Chao, S. Xiaojie, Z. Yutong, W. Zhengjie, L. Limin, W. Tao, Z. Luye, Z. Yang, Y. Qin, Z. Peirong, S. Lihong and Z. Qiurong p. 1089  abstract

LETTERS TO THE EDITOR

Synthesis and Optical Properties of the Conformationally Locked Diarylmethene Derivative of the GFP Chromophore

N. S. Baleeva, A. Yu. Smirnov and M. S. Baranov p. 1101  abstract

Halogen-Containing 4-Hydroxybenzylidene-Rhodanines as Fast Protein Fluorogens

A. I. Sokolov, N. S. Baleeva and M. S. Baranov p. 1105  abstract